GRP78-IN-3

In vial of 0.5 g net

TargetMol Chemicals Inc.

Product Overview

Product / Grade Name

GRP78-IN-3

Product Description

GRP78-IN-3, a potent small-molecule-competitive inhibitor of Hsp70 substrate binding and is a selective Grp78 (HSPA5) inhibitor with an IC50 of 0.59 μM. GRP78-IN-3 is 7-fold selective for HspA5 compared to HspA9 (IC50 of 4.3 μM) and >20-fold selective for HspA5 compared to HspA2 (IC50 of 13.9 μM).

Hazard Classification

  • UN Number

    :

  • IMGD Class

    :

  • Packing Group

    :

Visual Overview

Corporate Video